Home Tools
Log in
Cart

Search Result

Search Results for " transient receptor potential channels "

20

Compounds

Cat No. Product Name Synonyms Targets
T40042 Evifacotrep TRP/TRPV Channel
Evifacotrep is a short transient receptor potential channel 5 ( TRPC5 ) antagonist (WO2020061162, compound 100). Evifacotrep can be used for the research of neurological diseases.
T7177 Capsazepine Apoptosis , TRP/TRPV Channel
Capsazepine is an antagonist of TRPV1 receptor ( IC50 : 562 nM). Capsazepine blocks the painful sensation of heat caused by capsaicin (the active ingredient of chilli pepper) which activates the TRPV1 ion channel. It is ...
T2298 ML204 TRP/TRPV Channel
ML204 is a novel potent antagonist that selectively modulates native TRPC4/C5 ion channels.
T22124 Oleoyl Serotonin TRP/TRPV Channel
Oleoyl Serotonin is an antagonist of hTRPV1 with an IC50 of 2.57 μM.
T12514 Podocarpic acid Others , TRP/TRPV Channel
Podocarpic acid is a natural product and a novel TRPA1 activator.
T6848 GSK1016790A GSK101 Calcium Channel , TRP/TRPV Channel
GSK1016790A (GSK101) (GSK101) is a novel, potent activator of TRPV4 (transient receptor potential vanilloid 4) with EC50 of 34 nM in choroid plexus epithelial cells.
T6977 SB-366791 SB366791 TRP/TRPV Channel
SB-366791 is a new and selective cinnamide TRPV1 antagonist.
T6S1684 8-Gingerol Antioxidant , Antibacterial , TRP/TRPV Channel
1. 8-Gingerol has antioxidant activity. 2. 8-Gingerol has antimycobacterial activity. 3. 8-Gingerol could be used as an effective skin-whitening agent. 4. 8-Gingerol shows antipyretic and anti-inflammation characteristic...
T6617 Optovin TRP/TRPV Channel
Optovin is a TRPA1 activator, which is reversibly photoactivated.
T1814 ICILIN AG-3-5 TRP/TRPV Channel
ICILIN (AG-3-5) is a synthetic TRPM8 ion channel super-agonist.
T2807 Caffeic Acid Lipoxygenase , Endogenous Metabolite , TRP/TRPV Channel
Caffeic Acid is an orally bioavailable, hydroxycinnamic acid derivative and polyphenol, with potential anti-oxidant, anti-inflammatory, and antineoplastic activities.
T10537 BI-749327 TRP/TRPV Channel
BI-749327 is a high selectivity and orally bioavailable antagonist of TRPC6 (IC50s: 13 nM, 19 nM and 15 nM for mouse, human and guinea pig TRPC6).
T5698 TRPM8 antagonist 2 TRP/TRPV Channel
TRPM8 antagonist 2 is a potent and selective TRPM8 antagonist with an IC50 of 0.2 nM. TRPM8 antagonist 2 is used in the research of neuropathic pain syndromes.
T6660 SB-705498 TRP/TRPV Channel
SB705498 is a TRPV1 antagonist for hTRPV1. SB-705498 has been investigated for the treatment of Rhinitis, Chronic Cough, and Non-allergic Rhinitis.
T7430 AM-0902 TRP/TRPV Channel
AM-0902 is a potent and specific TRPA1 antagonist (IC50s: 71/131 nM for rTRPA1 and hTRPA1).
T16763 RN-1747 TRP/TRPV Channel
RN-1747 is a selective transient receptor potential cation channel subfamily V member 4 agonists (EC50: 0.77 μM, 4.0 μM, and 4.1 μM for hTRPV4, mTRPV4, and rTRPV4 respectively). RN-1747 also antagonizes TRPM8 (IC50: 4 μM...
T15628 JT010 TRP/TRPV Channel
JT010 is an effective agonist of TRPA1 (EC50 = 0.65 nM).
T9709 TRPM8 antagonist 3 TRP/TRPV Channel
TRPM8 antagonist 3 is a blocker of TRPM8 (IC50 = 11 nM).
T10300 AMG2850 TRP/TRPV Channel
AMG2850 is a potent, orally bioavailable, and selective antagonist of transient receptor potential melastatin 8 (TRPM8).
T5640 GSK2193874 TRP/TRPV Channel
GSK2193874 was identified as a selective, orally active TRPV4 blocker.
1 2 3 4 5
TargetMol